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Wednesday, February 17, 2010

Selected List of Medications approved by the AAP for use in breastfeeding mothers (AAP list revised 8/04)

Unlike women in general, pregnant and lactating mothers have dietary restrictions and also the necessity of consuming food. below we present a list of taboos and what should be consumed by pregnant women and lactating mothers
Generic nameTrade NameAAP approved?*Pregnancy Risk Category**Lactation Risk Category**
Analgesics (Pain-killers) [more]
AcetaminophenTylenolApprovedBL1
ColchicineColchicineApprovedDL4
NefopamAcupanApproved-NR
     Non-steroidal anti-inflammatory analgesics (NSAIDs) [more]
Azapropazone (apazone)RheumoxApproved-L2
Dipyrone (banned in the US & UK)-Approved-NR
Flufenamic acid-Approved-NR
IbuprofenAdvil, Nuprin, Motrin, PediaprofinApprovedB (1st, 2nd trim.)
D (3rd trim.)
L1
IndomethacinIndocinApprovedB (1st, 2nd trim.)
D (3rd trim.)
L3
KetorolacToradol, AcularApprovedB (1st, 2nd trim.)
D (3rd trim.)
L2
Mefenamic acidPonstan, PonstelApproved-NR
NaproxenAnaprox, Naprosyn, Naproxen, AleveApprovedBL3
L4 (for chronic use)
PhenylbutazoneButazolidineApproved-NR
PiroxicamFeldeneApprovedBL2
SuprofenProfenalApproved-NR
TolmetinTolectinApprovedCL3
     Narcotic analgesics [more]
ButorphanolStadolApprovedB (1st, 2nd trim.)
D (3rd trim.)
L3
CodeineTylenol #3, #4ApprovedCL3
FentanylSublimazeApprovedBL2
MeperidineDemerolApprovedBL2
L3 (if used early postpartum)
MethadoneDolophineApprovedBL3
MorphineMorphineApprovedBL3
PropoxypheneDarvocet N, Propacet, DarvonApprovedCL2
Anesthesia, Anesthetics [more][contents]
HalothaneFluothaneApprovedCL2
LidocaineXylocaineApprovedCL2
MethohexitalBrevitalApprovedBL3
ThiopentalPentothalApprovedCL3
Antacids, GI meds[contents]
Cimetidine (Antacid)TagametApprovedBL2
Cisapride (GI tract stimulant)PropulsidApprovedCL2
Domperidone (used for nausea & vomiting, stimulates lactation) [more]MotilumApproved-L1
Antibiotics[contents]
AmoxicillinLarotid, AmoxilApprovedBL1
AztreonamAzactamApprovedBL2
CefadroxilUltracef, DuricefApprovedBL1
CefazolinAncef, KefzolApprovedBL1
CefotaximeClaforanApprovedBL2
CefoxitinMefoxinApprovedBL1
CefprozilCefzilApprovedCL1
CeftazidimeCeftazidime, Fortaz, TaxidimeApprovedBL1
CeftriaxoneRocephinApprovedBL2
Ciprofloxacin [more]CiproApprovedCL3
ClindamycinCleocinApprovedBL3
ErythromycinE-Mycin, Ery-tab, ERYC, IlosoneApprovedBL1
L3 early postnatal
Fleroxacin-Approved-NR
GentamicinGaramycinApprovedCL2
KanamycinKebecil, KantrexApprovedDL2
MoxalactamMoxamApproved-NR
NitrofurantoinMacrobidApprovedBL2
OfloxacinFloxinApprovedCL2
Penicillin-ApprovedBL1
StreptomycinStreptomycinApprovedDL3
Sulbactam-Approved-NR
SulfisoxazoleGantrisin, Azo-GantrisinApprovedCL2
TetracyclineAchromycin, Sumycin, TerramycinApprovedDL2
TicarcillinTicarcillin, Ticar, TimentinApprovedBL1
Trimethoprim/sulfamethoxazoleProloprim, TrimpexApprovedCL3
Anticoagulants[contents]
Bishydroxycoumarin (dicumarol)-Approved-NR
WarfarinCoumadin, PanwarfinApprovedDL2
Anticonvulsants[contents]
CarbamazepineTegretol, EpitolApprovedCL2
EthosuximideZarontinApprovedCL4
Magnesium sulfateEpsom saltApprovedBL1
PhenytoinDilantinApprovedDL2
Valproic acidDepakene, DepakoteApprovedDL2
Antifungals[contents]
Fluconazole [more]DiflucanApprovedCL2
KetoconazoleNizoral Shampoo, NizoralApprovedCL2
Antihistamines [more][contents]
Dexbrompheniramine maleate with d-isoephedrine-Approved-NR
FexofenadineAllegraApprovedCL2
LoratadineClaritinApprovedBL1
TerfenadineSeldaneApproved-NR
TriprolidineActidil, ActifedApprovedCL1
Antivirals[contents]
Acyclovir [more]ZoviraxApprovedCL2
Interferon-alpha [more]Alferon N, Interferon AlphaApprovedCL2
Arthritis meds (see also: pain meds)[contents]
Gold saltsRidaura, Myochrysine, SolganalApprovedCL5
Asthma meds (see also: steroids)[contents]
DyphyllineDilor, Lufyllin, DyphyllineApprovedCL3
TerbutalineBricanyl, BrethineApprovedBL2
TheophyllineAminophylline, Quibron, Theo-DurApprovedCL3
Contraceptives, Hormones [more][contents]
EstradiolEstratab, Permarin, MenestApprovedXL3 (may interfere with milk production)
Clogestone-Approved-NR
Contraceptive pill with estrogen/progesteronePreven, Seasonale, Norinyl, Norlestin, Ortho-Novum, Ovral, Lunelle injection, Ortho-Evra patch, etc.ApprovedXL3 (may interfere with milk production)
LevonorgestrelNorplant, Mirena, Plan BApprovedXL2
MedroxyprogesteroneProvera, Depo-Provera, CycrinApprovedDL1
L4 (if used first 3 days postpartum)
NorethynodrelEnovidApprovedXL2
ProgesteroneCrinone, PrometriumApproved-L3
Cough meds [more][contents]
CodeineTylenol #3, #4ApprovedCL3
Noscapine-Approved-NR
Decongestants [more][contents]
PseudoephedrineSudafed, Halofed, Novafed, ActifedApprovedCL3 (for acute use)
L4 (for chronic use)
Diabetes meds[contents]
Note: Insulin has not been reviewed by the AAP. Pregnancy risk category = B; Lactation risk category = L1.
TolbutamideOramide, OrinaseApprovedDL3
Diarrhea meds[contents]
LoperamideImodium, Pepto Diarrhea Control, Maalox Antidiarrheal Caplets, Kaopectate II Caplets, Immodium AdvancedApprovedBL2
** Note: Pepto-Bismol & Kaopectate (bismuth subsalicylate is the active ingredient in both) are not recommended for routine use by nursing moms, due to the association of salicylates with Reyes syndrome in children. [more]
Diuretics[contents]
AcetazolamideDazamide, DiamoxApprovedCL2
BendroflumethiazideNaturetinApprovedDL4 (may inhibit lactation)
ChlorothiazideHydrodiurilApprovedDL3
ChlorthalidoneHygrotonApprovedDL3
HydrochlorothiazideHydrodiuril, Esidrix, OreticApprovedDL2
SpironolactoneAldactoneApprovedDL2
Galactagogues (milk supply) [more][contents]
DomperidoneMotilumApproved-L1
Heart, Blood Pressure meds 
(Antiarrhythmics, Antihypertensives, Cardiac stimulants)
[contents]
     Antiarrhythmics
DisopyramideNorpace, NapamideApprovedCL2
FlecainideTambocorApprovedCL3
MexiletineMexitilApprovedBL2
ProcainamidePronestyl, ProcanApprovedCL3
QuinidineQuinaglute, QuinidexApprovedCL2
     Antihypertensives
CaptoprilCapotenApprovedDL3 (if used after 30 days)
Diltiazem/Diltiazem HCLCardizem Sr, Dilacor-XR, Diltiazem, Cardizem CDApprovedCL3
Enalapril/Enalapril MaleateVasotecApprovedC (1st trim.)
D (2nd, 3rd trim.)
L2
HydralazineApresolineApprovedCL2
LabetalolTrandate, NormodyneApprovedCL2
MethyldopaAldometApprovedCL2
MetoprololToprol XL, LopressorApprovedBL3
MinoxidilLoniten, Minodyl, RogaineApprovedCL2(topically)
L3 (orally)
NadololCorgard, NadololApprovedCL4
NifedipineAdalat, ProcardiaApprovedCL2
OxprenololApsolox, Slow-Trasicor, TrasicorApproved-NR
PropranololInderolApprovedCL2
SotalolBetapaceApprovedBL3
TimololBlocadrenApprovedCL2
VerapamilCalan, Isoptin, Covera-HSApprovedCL2
     Cardiac stimulants
DigoxinLanoxin, LanoxicapsApprovedCL2
Laxatives [more][contents]
Cascara/Cascara Sagrada-ApprovedCL3
Danthron-Approved-NR
Magnesium sulfateEpsom saltApprovedBL1
Senna-Approved-L3
Malaria meds[contents]
ChloroquineAralen, Novo-chloroquineApprovedCL3
HydroxychloroquinePlaquenilApprovedCL2
PyrimethamineDaraprimApprovedCL4
QuinineQuinammApprovedDL2
Medical Testing [more][contents]
Diatrizoate-Approved-NR
Fluorescein-ApprovedCL3
Gadopentetic (Gadolinium)-ApprovedCL2
IohexolOmnipaqueApprovedBL2
Iopanoic acidTelepaqueApprovedDL2
MetrizamideAmipaqueApprovedBL2
MetrizoateIsopaqueApprovedBL2
Migraine meds (see also: pain meds) [more][contents]
SumatriptanImitrexApprovedCL3
Sedatives [more][contents]
Chloral hydrateAquachloral, NoctecApprovedCL3
Methyprylon (withdrawn from use in US & Canada)-Approved-NR
Bromide-ApprovedDL5
SecobarbitalSeconalApprovedDL3
Sleep Aids[contents]
Zolpidem/Zolpidem TartrateAmbienApprovedBL3
Steroids[contents]
Methylprednisolone
[PDF high dosage methylprednisolone]
Solu-Medrol, Depo-Medrol, MedrolApprovedCL2
Prednisolone-ApprovedCL2
PrednisoneDeltasone, Meticorten, OrasoneApprovedCL2
Thyroid meds [more][contents]
Carbimazole-ApprovedDL3
Methimazole (active metabolite of carbimazole)TapazoleApprovedDL3
PropylthiouracilPTUApprovedDL2
Thiouracil-Approved-NR
LevothyroxineSynthroid, Levothroid, Thyroid, Levo-T, LevoxylApprovedAL1
Tuberculosis meds[contents]
CycloserineSeromycinApprovedCL3
EthambutolEthambutol, MyambutolApprovedBL2
IsoniazidINH, LaniazidApprovedCL3
RifampinRifadin, RimactaneApprovedCL2
Vitamins [more][contents]
B-1 (thiamin)-Approved-NR
B-12 (Cyanocobalamin)-ApprovedAL1
B-6 (pyridoxine)-ApprovedAL2L4 in high doses (may inhibit lactation)
D, vitaminCalciferol, Delta-dApprovedAL3 (do not overdose)
Folic acid-ApprovedA (1st, 2nd trim.)
C (3rd trim.)
L1
K-1, vitamin (Phytonadione)-ApprovedCL1
Riboflavin/B2 -ApprovedAL1
Miscellaneous[contents]
Acitretin (Anti-psoriasis)SoriataneApproved-NR
Alcohol/Ethanol [more]-ApprovedDL3
AllopurinolZyloprim, LopurinApprovedCL2
Antimony-Approved-NR
Atropine (Anticholinergic, drying agent)Belladonna, AtropineApprovedCL3
Azapropazone/apazone (Antirheumatic)RheumoxApproved-L2
Baclofen (muscle relaxant)Lioresal, AtrofenApprovedCL2
Barbiturate-Approved-NR
Caffeine [more]Vivarin, NoDoz, CoffeeApprovedBL2
Carbetocin (Antihemorrhagic)DuratocinApproved-NR
Chloroform-Approved-NR
Cisplatin (Anti-cancer)PlatinolApprovedDL4
Dapsone (Antileprosy)Avlosulfon, DDSApprovedCL4
Hydroxychloroquine (Antirheumatic, lupus)PlaquenilApprovedCL2
Iodides-Approved-NR
Iodine-Approved-NR
Iodine (povidone-iodine, eg, in a vaginal douche)-Approved-NR
Ivermectin (Antiparasitic)MectizanApprovedCL3
Nalidixic acid (Urinary Anti-infective)NegGramApprovedBL4
Norsteroids-Approved-NR
Pyridostigmine (Muscle stimulant)Mestinon, RegonolApprovedCL2
Scopolamine (Motion sickness)Transderm ScopeApprovedCL3
SulfapyridineDagenanApproved-NR
Timolol (glaucoma med)BlocadrenApprovedDL3


*  Per the AAP Policy Statement The Transfer of Drugs and Other Chemicals Into Human Milk, revised September 2001.

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